Silica sulfuric acid promotes aza-Michael addition reactions under solvent-free condition as a heterogeneous and reusable catalyst.

نویسندگان

  • Yan Wang
  • Yan-Qin Yuan
  • Sheng-Rong Guo
چکیده

A highly efficient, inexpensive, recyclable, convenient, and green protocol for chemoselective aza-Michael addition reactions of amines/thiols to alpha,beta-unsaturated compounds using silica sulfuric acid (SSA or SiO(2)-SO(3)H) was developed. This method is simple, convenient and the title compounds are produced in good to excellent yields.

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عنوان ژورنال:
  • Molecules

دوره 14 11  شماره 

صفحات  -

تاریخ انتشار 2009